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Palladium-Catalyzed α-Stereoselective O-Glycosylation of O(3)-Acylated Glycals
, M.C. Galan
Published in American Chemical Society
2017
PMID: 28514163
Volume: 19
   
Issue: 11
Pages: 2857 - 2860
Abstract
Pd(MeCN)2Cl2 enables the α-stereoselective catalytic synthesis of 2,3-unsaturated O-glycosides from O(3)-acylated glycals without the requirement for additives to preactivate either donor or nucleophile. Mechanistic studies suggest that, unlike traditional (η3-allyl)palladium-mediated processes, the reaction proceeds via an alkoxy-palladium intermediate that increases the proton acidity and oxygen nucleophilicity of the alcohol. The method is exemplified with the synthesis of a range of glycosides and glycoconjugates of synthetic utility. © 2017 American Chemical Society.
About the journal
JournalData powered by TypesetOrganic Letters
PublisherData powered by TypesetAmerican Chemical Society
ISSN15237060